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Publications

2021年

2021年

◾️学術論文/学会誌

Nobel bicyclic pyrazoles as potent ALK2 (R206H) inhibitors for the treatment of fibrodysplasia ossificans progressiva

Yamamoto H., Sakai N., Ohte S., Sato T., Sekimata K., Matsumoto T., Nakamura K., Watanabe H., Mishima-Tsumagari C., Tanaka A., Hashizume Y., Honma T., Katagiri T., Miyazono K., Tomoda H., Shirouzu M., Koyama H.

Bioorg. Med. Chem. Lett. Online ahead of print (2021).

Inhibitory effects of sesquiterpene lactones from the Indonesian marine sponge Lamellodysidea cf. herbacea on bone morphogenetic protein-induced osteoblastic differentiation.

Ohte S., Yamazaki H., Takahashi O., Rotinsulu H., Wewengkang DS., Sumilat DA., Abdjul DB., Maarisit W., Kapojos MM., Zhang H., Hayashi F., Namikoshi M., Katagiri T., Tomoda H., Uchida R.

Bioorg. Med. Chem. Lett. 35, 127783 (2021).

抗真菌薬活性増強剤の開拓

小林 啓介、内田 龍児、福田 隆志、長光 亨、長井 賢一郎、供田 洋 

化学工業 72, 28-37 (2021).

◾️学会発表

2022

2022

Discovery of prescopranone, a key intermediate in scopranone biosynthesis
Demachi A., Ohte S., Uchida R., Shin-ya K., Ohshiro T., Tomoda H., Ikeda H.
J. Antibiot. 75, 305-311 (2022).

Kimidinomycin, a new antibiotic against Mycobacterium avium complex, produced by Streptomyces sp. KKTA-0263

Hikima A., Asamizu S., Onaka H., Zhang H., Tomoda H., Koyama N.
J. Antibiot. 75, 72-76 (2022).

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