Screening for Small Molecule Inhibitors of BMP-Induced Osteoblastic Differentiation from Indonesian Marine Invertebrates.

Yamazaki H., Ohte S., Rotinsulu H., Wewengkang DS., Sumilat DA., Abdjul DB., Maarisit W., Kapojos MM., Namikoshi M., Katagiri T., Tomoda H., Uchida R.

Mar. Drugs 18, 606 (2020).

 

Evaluation of Anti-Mycobacterial Compounds in a Silkworm Infection Model with Mycobacteroides abscessus

Hosoda K., Koyama N., Hamamoto H., Yagi A., Uchida R., Kanamoto A., Tomada H. 

Molecules 25, E4971 (2020).

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Quantitative analysis of selective glycosylation of saccharides with aromatic amines

Hanai T., Shimada K., Koyama N., Nohara Y. 

Carbohydr. Res. 498, 108171 (2020).

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Discovery of oosporein as a new inhibitor of influenza virus cap-snatching activity

Koyama N., Shibagaki Y., Okuwaki M., Hattori S., Tomoda H. 

Int. J. Pharm. Sci. Res. 7, 137 (2020).

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Penicillic acid congener, a new inhibitor of BMP-induced alkaline phosphatase activity in myoblasts, produced by the fungus Penicillium sp. BF-0343

Koyama N., Otoguro Y., Ohte S., Katagiri T., Tomoda H. 

Nat. Prod. Communum. 15, 1-5 (2020)

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Steffimycin E new anti-mycobacterial agent against Mycobacterium avium complex, produced by Streptomyces sp. OPMA02852.

Koyama N., Shigeno S., Kanamoto A., Tomoda H. 

J. Antibiot. 73, 581-584 (2020).

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2-Epi-anthracimycin, a new cytotoxic agent from the marine-derived actinomycete Streptomyces sp. OPMA00631. 

Fukuda T., Nagai K., Kanamoto A., Tomoda H.

J. Antibiot. 73, 548-553 (2020).

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A new diketopiperazine-like inhibitor of bone morphogenetic protein-induced osteoblastic differentiation produced by marine-derived Aspergillus sp. BFM-0085. 

Ohte S., Shiokawa T., Koyama N., Katagiri T., Imada C., Tomoda H. 

J. Antibiot. 73, 554-558 (2020).

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New Terpendole Congeners, Inhibitors of Sterol O-Acyltransferase, Produced by Volutella citrinella BF-0440.

Nur EAA., Kobayashi K., Amagai A., Ohshiro T., Tomoda H. 

Molecules 25, 3079 (2020).

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Synthesis and Absolute Configuration of Habiterpenol.

Konya M., Shimoyama K., Arima S., Fukuda T., Uchida R., Tomoda H., Nagamitsu T.

Org. Lett. 22, 5131-5134 (2020).

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The Anti-atherogenic Activity of Beauveriolide Derivative BVD327, a Sterol O-Acyltransferase 2-Selective Inhibitor, in Apolipoprotein E Knockout Mice.

Ohshiro T., Imuta S., Hijikuro I., Yagyu H., Takahashi T., Doi T., Ishibashi S., Tomoda H. 

Biol. Pharm. Bull. 43, 951-958 (2020).

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Voluhemins, new inhibitors of sterol O-acyltransferase, produced by Volutella citrinella BF-0440.

Ohshiro T., Morita H., Nur EAA., Hosoda K., Uchida R., Tomoda H. 

J. Antibiot. 73, 748-755 (2020).

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Inhibition of cholesteryl ester synthesis by polyacetylenes from Atractylodes rhizome.

Nur EAA., Ohshiro T., Kobayashi K., Wu J., Wahyudin E., Zhang H., Hayashi F, Kawagishi H, Tomoda H. 

Bioorg. Med. Chem. Lett. 30, 126997 (2020).

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Polyketide glycosides phialotides A to H, new potentiators of amphotericin B activity, produced by Pseudophialophora sp. BF-0158. 

Yagi A., Uchida R., Kobayashi K., Tomoda H. 

J. Antibiot. 73, 211-223 (2020).